home Audience 4 Instructions for use and description of the medicine validol. Liquid validol instructions for use

Instructions for use and description of the medicine validol. Liquid validol instructions for use

For “heart” ailments, “nerves” and poor health, white tablets with a sharp menthol taste - validol - have been kept in the home medicine cabinet for many years. Indications for the use of this medicine include both pain in the heart area and stress and hysteria. In what cases should you resort to such “first aid”?

What does validol help with?

1. Validol is used in complex therapy as an antianginal agent

We are talking about stopping the attack angina pectoris. Angina is a condition in which pain occurs behind the sternum and in the region of the heart, radiating to the back under the shoulder blade. A person feels a lack of air, tightness in the chest and uncontrollable anxiety associated with this.

The cause of angina is insufficient oxygen supply to the heart muscle. Since attacks are fraught with the development of myocardial infarction, they must be stopped at an early stage. For these purposes, validol is used, among other things.

Unlike nitroglycerin, which increases the amount of oxygen delivered to the heart and at the same time reduces the need for it, validol is classified as a coronary dilator. It is suitable for preventing mild attacks in the initial stages.

However, in case of a real heart attack, you should not rely on the help of validol. It “distracts” from the problem in which it is necessary to urgently call the ambulance. In any case, instead of self-medicating, you need to go to a cardiologist and find out the true causes of pain in the heart area.

2. Validol slightly lowers blood pressure during stress and nervous tension

It is impossible to cure arterial hypertension with the help of tablets or capsules; it will be possible to stabilize the pulse and calm down by expanding the lumen of blood vessels and stimulating the receptors responsible for the production of endorphin.

The tablets have a mild analgesic effect. Taking validol should be combined with the elimination of factors that increase blood pressure: mental and physical stress, negative emotions, sleep disorders.

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3. Treatment of neuroses

This form of mental stress is not considered a pathology, but, nevertheless, prevents a person from leading a full life. In addition to manifestations from the nervous system, somatics makes itself felt:

Heart rate increases
Sweating increases
Loss of appetite (loss or excessive absorption of food)
Suffering from insomnia or drowsiness at any time of the day
There is irritability, tearfulness
Headaches and migraines appear
Attention becomes distracted and inadequate reactions to what is happening occur.

Hysteria is complemented by movement disorders, loss of vision, hearing, voice, inappropriate behavior, loss of orientation in space and time.

Validol expands the lumen of blood vessels, has a sedative effect and is used as part of complex therapy.

4. Validol during pregnancy

Validol is prescribed during pregnancy for:

Relief of angina attacks
Soothing headaches, migraines
As a detoxifier (this property can be used to combat motion sickness and motion sickness)
To lower blood pressure

You should remember about possible side effects and contraindications; self-medication can be dangerous, so before taking the drug during pregnancy, you should consult your doctor.

5. Inhalations for dry cough

Help alleviate the patient's condition. Menthol helps eliminate swelling of the mucous membrane, improves microcirculation and facilitates mucus discharge, and softens the throat.

To prepare the solution, bring 0.5 liters of water to a boil, add 5-7 drops of iodine, 1 tsp. baking soda and crushed tablet. Breathe over the pan or through the spout of the teapot for 10 minutes.

For children, do not add soda and iodine to the cough solution in the water; use only validol, 1 tablet per 1 liter of water.

6. Add to drops for a runny nose

The tablet is dissolved in water and mixed with drops or nasal spray based on sea water. Menthol helps ease breathing and relieves nasal congestion.

Before being treated in this way, you should make sure that you are not allergic to the components of the drug. Validol or Corvalol can be used as a medicine.

Does validol help with a hangover?

The compatibility of validol and alcoholic beverages is a big question. After alcohol, it is better not to use the drug as a drug to help get rid of morning sickness, headaches, confusion and general malaise. Pharmacology offers a number of drugs with an anti-hangover effect; validol is not on this list.

How to take validol tablets

The instructions give clear instructions in this regard: both “for the heart” and “for the nerves” the drug is taken sublingually - under the tongue until completely dissolved.

Similarly, glycine and other drugs are taken that irritate the oral mucosa and are absorbed into the blood. It is for this reason that the drug begins to act quite quickly - relief occurs within a few minutes after administration.

How many tablets can you take per day?

Simultaneous use involves dissolving one or two tablets, however, in order not to cause harm to the body, the daily dose should not exceed 4 tablets.

If the attack cannot be relieved with the indicated dose, your health worsens, chest pain increases and there is not enough air, you should immediately seek medical help, a pre-infarction condition may develop.

There is another form of release of validol - in drops. A single dosage is 5-6 drops, the medicine is dripped onto a cube of refined sugar and placed under the tongue.

An overdose threatens to intoxicate the body and is expressed in:

Inhibition of the functions of the central nervous system - lethargy, apathy, weakness, lethargy, drowsiness;
Lacrimation, since menthol provokes irritation of the lacrimal glands;
Nausea or vomiting (this is how the body tries to get rid of excess harmful substances)

Side effects occur in a similar way. In addition, hypotension and an allergy to the components of the drug may develop. That is why the list of contraindications includes low blood pressure and individual intolerance to the drug.

Analogues of the drug

The benefits of validol are enhanced by additional substances added to the drug. Validol with glucose, among other things, enhances metabolism and stimulates redox processes in the body. This drug should be taken with extreme caution by people suffering from diabetes.
The following drugs are also used as part of complex therapy:

Can validol be taken with other medications?

Validol and its analogues enhance the effect of sedatives, antihypertensive and neurotropic drugs, but before combining them, you should consult your doctor.

During treatment, you may experience absent-mindedness, inattention, and drowsiness, so you should not drive or take on responsible tasks that require full concentration.

Numerous reviews indicate the reliability of this affordable drug, proven over the years. People with heart problems, autonomic dysfunction and mental disorders should carry validol with them as first aid.

Validol
Instructions for medical use - RU No. P N015115/01

Last modified date: 15.06.2017

Dosage form

Sublingual capsules.

Compound

1 capsule contains:

Active components:

Levomenthol solution in menthyl isovalerate (validol) - 100 mg.

Composition of the shell of gelatin capsules:

pharmaceutical gelatin, glycerol, methyl parahydroxybenzoate, propyl parahydroxybenzoate, purified water.

Description of the dosage form

Soft gelatin capsules, spherical, light yellow in color.

The contents of the capsules are a clear, colorless or slightly colored oily liquid with a menthol odor.

Pharmacological group

Coronodilating agent of reflex action.

Pharmacodynamics

It has a sedative effect and has a moderate reflex vasodilator effect due to irritation of sensitive nerve endings. Stimulates the production and release of enkephalins. endorphins and a number of other peptides, kinins (due to irritation of mucosal receptors), which take an active part in the regulation of vascular permeability and the formation of pain.

Pharmacokinetics

When administered sublingually, it is absorbed from the oral mucosa. After absorption, it is biotransformed in the liver and excreted by the kidneys in the form of glucuronides.

Indications

Functional cardialgia, neuroses, and also as an antiemetic for sea and air sickness.

Contraindications

Hypersensitivity to the components of the drug.

Directions for use and doses

Validol is prescribed to adults under the tongue. The capsule should be kept in the mouth under the tongue until completely absorbed. Take 1 capsule 2-3 times a day.

The daily frequency and duration of administration is determined depending on the effectiveness of treatment. If the effect is not sufficiently pronounced or when some patients do not experience an effect within the next 5 minutes after taking the drug, it is necessary to contact your doctor to prescribe another therapy.

Side effects

With long-term use of validol, mild nausea, dizziness, and lacrimation may occur. These phenomena usually go away on their own.

Overdose

Symptoms:

headache, nausea, agitation, cardiac dysfunction, decreased blood pressure, depression of the central nervous system.

Treatment:

stop the drug. Symptomatic therapy.

Interaction

When used together with drugs that depress the central nervous system, it enhances the inhibitory effect of the latter.

The simultaneous use of Validol with nitrates reduces the headache that occurs when using them.

Release form

Sublingual capsules 100 mg.

10 capsules in a blister pack, 2 blister packs each along with instructions for use in a cardboard box.

Storage conditions

In a dry place, protected from light, at a temperature of 15 to 25 ° C.

Keep out of the reach of children.

Almost every one of us has a first aid kit at home with the necessary drugs to maintain optimal well-being. We often even take the most necessary medications that help in various unforeseen situations with us in our purse. To be aware of which drug will often help you, find out more information about such a useful and sometimes irreplaceable drug as Validol: indications for its use, whether it has side effects, whether it has analogues.

Composition and mechanism of action of the drug

Menthol solution in menthyl isovalerate is the international name of the drug. Without going into complex medical formulas, the active ingredients are menthol, which is made from peppermint leaves, and isovaleric acid, an extract from valerian root. Validol works like this: the nerve endings of the mucous membrane receptors react to menthol, as a result of which the body produces substances that can relieve pain and produce a calming effect. The medicine is not accumulated by the body, cases of overdose are very rare.

People diagnosed with hypertension are often interested in the question: Does Validol lower or increase blood pressure? This is a vasodilator, therefore, according to the laws of physics, since the lumen of the blood vessels increases after taking the medicine, the blood pressure in them decreases. But according to pharmaceutical standards, Validol is not defined as an independent drug that reduces blood pressure. For this purpose, it can be prescribed only in complex therapy, as an adjuvant.

Release form

The drug is available in the following dosage forms:

Tablets are the most widely used option. The composition of Validol tablets includes 60 mg of validol and excipients: sugar or powdered sugar, calcium stearate.
Capsules are made without the use of sugar and use a gelatin shell. Validol in capsules can be in a dosage of 50 ml or 100 ml of the active substance.
Drops - this liquid form is an alcohol solution, oily in appearance, with a strong menthol odor.

Due to its accessibility and wide scope of application, it is imperative to pay attention to whether a particular drug contains sugar, because Validol with glucose is prohibited from being used for treatment by people with diabetes. For them, the best option in most cases will be capsules, although some manufacturers have now started producing Validol tablets without sugar.

What does Validol help with: indications for use

The drug is prescribed for the following conditions:

neuroses – when a person’s psyche is overstrained for a long time due to mental or emotional overload;
hysteria - manifested by fits of uncontrollable laughter, crying, screaming, etc.;
cardialgia – pain manifested in the heart area;
angina pectoris (in such cases, Validol is combined with Nitroglycerin, because Validol alone does not relieve spasm of the heart muscle, but only relieves pain);
nausea and motion sickness in transport, with seasickness;
with high blood pressure as part of complex treatment.

Instructions for use and dosage

Many people are interested in the question, how to take Validol correctly - only when feeling unwell or in a course? We emphasize that only a doctor should prescribe long-term treatment. This medicine is characterized by the fact that it works within 5 minutes, and if there is no improvement, you should seek additional medical help. Let's outline the application diagrams:

tablets or capsules – 1 pc. sublingually, under the tongue until completely absorbed, no more than 3 times a day;
drops are applied to a piece of sugar and dissolved, 3-6 drops at a time, the daily dose is no more than 24 drops in 4 doses.

Side effects and contraindications

After taking Validol, no side effects occur, with the exception of individual intolerance to the components of the drug. Very rarely, nausea, dizziness, and lacrimation are observed, which quickly disappear without the use of any additional measures. With prolonged use of the medicine, allergic reactions may intensify, so the course of treatment should always be taken under the supervision of a doctor. Validol should not be taken with alcohol, and the effectiveness of this hangover reliever, as is often discussed, has not been proven.

Validol is prescribed with caution during pregnancy, because menthol can provoke contraction of the smooth muscles of the uterus, which leads to a threat to pregnancy. Women during breastfeeding can similarly take this drug only as prescribed by a doctor if the potential benefits outweigh the risk factors for the child. This medicine is not used in children under 12 years of age. Finally, do not forget that the drug is contraindicated for low blood pressure.

Analogues of the drug Validol

The following drugs have similar properties and indications for use:

Corvalment - capsules based on menthol and isovaleric acid, dilate blood vessels and have a calming effect.
Corvalol, Valocordin - similar in their calming effect, they contain peppermint oil.
Valoserdin - available in the form of drops, the main active ingredient is phenobarbital, contains peppermint oil as an auxiliary component. It has a calming and mild hypnotic effect, relieves pain in the heart area. They differ in a number of contraindications.

Where to buy and how much it costs

Today, many pharmacies offer their services to us. To purchase Validol profitably, you need to know how much the drug costs at different points of sale. In Moscow, St. Petersburg and other big cities of Russia, you can conveniently order medicine through online pharmacies with delivery, saving your time. For example, let’s compare information on some points of sale in Moscow.

Validol is a drug that has a reflex vasodilator effect. The medicine is used as part of combination antianginal therapy, as well as for the treatment of a number of other diseases. The drug is available in the following dosage forms:

Validol drops;
Validol capsules;
Validol tablets.

1 tablet of Validol contains 60 mg of menthol solution in isovaleric acid menthol ester. The drug is dispensed without a doctor's prescription.

Pharmacological action of Validol

According to the instructions, Validol produces moderate reflex vasodilator and sedative (calming effect on the central nervous system) effects. The mechanism of action of the drug is based on reflex reactions associated with irritation of sensitive nerve endings. The properties of Validol are close to menthol. Due to irritation of mucous surface receptors by the active component, endorphins, enkephalins, peptides and dynorphins are released, which play a critical role in regulating pain, the permeability of vascular walls and other processes in the human body. Also, during such reactions, other physiologically active compounds are released, such as kinins, histamine and others. The clinical effect is observed 5 minutes after sublingual application of Validol.

Indications for use of Validol

According to the instructions, Validol is prescribed for such conditions and diseases as:

neuroses;
attacks of angina (as part of combination therapy);
hysterical states, hysteria;
functional cardialgia, neurocirculatory dystonia of the cardiac type;
sea and air sickness (as an antiemetic).

Directions for use and dosage

Validol tablets are taken orally, but are not swallowed whole, but placed under the tongue until completely dissolved, that is, sublingually. The dosage is 1 tablet 2-3 times a day. The duration of treatment is determined depending on the effectiveness of the drug for a particular patient. This means that if after taking the drug the therapeutic effect does not occur within 5-10 minutes, then it is advisable to use other medications.

Validol in drops is taken 3 drops at a time, and the drug must be dripped onto sugar and kept in the mouth until completely dissolved. The daily dose of the drug should not exceed 9-24 drops, depending on the disease and condition of the patient. Frequency of administration – 3-4 times during the day. If necessary, the dosage is increased.

Validol in capsules is taken in the same doses as in tablets, that is, 1 piece twice a day, but the exact dosage is adjusted by a doctor. Capsules must be kept under the tongue.

Side effects of Validol

As a result of taking Validol, the following reactions from the body can sometimes occur:

mild nausea;
lacrimation;
dizziness.

If such symptoms occur, there is no need for symptomatic treatment, because such phenomena go away on their own.

Contraindications for use

The drug is contraindicated in case of individual intolerance to its components, acute myocardial infarction and severe hypotension. Validol should be prescribed with caution during pregnancy and lactation. When treated with this drug, constant medical monitoring of the condition of the mother and fetus is required. During pregnancy, Validol can be prescribed only for special medical reasons.

When taking the medicine in the dosages specified in the instructions, there are no disturbances in concentration and other mental reactions, therefore it is allowed to drive vehicles and other mechanisms during therapy.

The drug is not prescribed to children, since its effect on this group of patients has not been studied.

Since the drug does not contain sugar, it can be taken by patients with diabetes, but without adding sugar as an excipient (when taking drops).

Conditions and shelf life

Validol should be stored in a cool, dark place in a well-closed container. The shelf life of tablets is 1.5 years, solution – 4 years, capsules – 2 years.

What is the drug for and what is it made of? How often can it be used? What exactly is Validol taken for? The drug is indicated for use in the following cases:

for the therapeutic treatment of angina pectoris;
with neurocircular dystonia;
nervous disorders of various types;
as an antiemetic for motion sickness.

Validol tablets are taken by holding them under the tongue until completely dissolved. Thus, you can use no more than 3 tablets per day. "Validol" capsules are drunk no more than 4 times a day. The dose for adults is no more than 2 units of tablets or capsules, and the daily dose should not exceed 4. In exceptional cases, the intake of Validol in capsules is increased.

Manufacturers produce the medicine "Validol" in 20 pieces per package, if these are capsules, and in tablets - 6 or 10 pieces weighing 60 mg.

Validol tablets contain the following chemical ingredients:

About 5% natural menthol or mint extract. In terms of content, 1 tablet contains 0.06 milligrams of the substance.
Excipients are used as excipients to impart flavor characteristics to the medicine. This is a powder made from sugar and calcium stearate.

The color of the tablets is crystal white or slightly yellowish. The shape is a flat cylinder, and there is a chamfer in the middle. The smell is quite strong, menthol. During production, inclusions of a gray tint and a coating of white powder are allowed.

Advantages of the drug

The use of Validol internally promotes vasodilation and also has a calming effect on the nervous system, while the patient does not fall asleep. Validol contains components that help improve blood circulation and reduce pain.

In general, this drug resembles menthol in its taste properties. The action of "Validol" is associated with reflex functions of the body or with an impact on nerve endings.

This effect occurs when:

stimulation of pain and the formation of enkephalins;
interaction between cells of the nervous and immune systems;
substances capable of producing particles to reduce headaches;
peptides that play a role in regulating pain;
vascular patency;
other metabolic processes.

Using the drug internally causes the release of some active components, such as kinin and histamine. After taking the medicine, you can feel the result after 5 minutes. The components included in the medicine partly remain inside the liver, and other products are excreted in the feces. The composition of the product does not change when excreted in urine or air.

In what cases should you not take the drug?

The instructions for use also stipulate cases in which taking the medicine is impossible.

These include:

intolerance to both individual components and the complex of ingredients contained;
low blood pressure;
initial stage of heart attack;
failure to reach adulthood.

The use of Validol when driving should be carried out with extreme caution. Also, you should not get carried away with it when doing work that requires special attention. Side effects such as dizziness and the desire to sleep cannot be excluded. How to take the product during pregnancy? The answer to this question can be obtained from your attending physician. As a rule, he prescribes taking a medicine in cases where the effectiveness of taking the medicine may exceed the risk for the birth of a future person. But these are only exceptional measures.

If it is not possible to lower blood pressure and, for example, pain in the chest area does not go away, then you need to act in other ways. To relieve high blood pressure, you need to use combination therapy. For this purpose, nitrates are additionally prescribed.

The indications for the use of Validol also have this important property: the drug cannot be prescribed to people with diabetes mellitus, since the drug also contains sweet foods.

Adverse events after taking the medicine

What Validol helps with has already been discussed above, but the question arises, does this product have side effects?

The instructions for use of Validol, along with the positive effects, also describe side effects:

feelings of nausea;
possible dizziness;
increased secretion of tears.

There is no need to take special measures to eliminate these factors. They will gradually pass without the help of doctors.

Does Validol increase or decrease blood pressure? This primarily depends on the patient’s health status.

When the product interacts with other drugs

It is possible that some actions of the drug may be enhanced when taking other medications concomitantly. But it is possible that there are cases of incompatibility of such solutions.

List of possible interactions:

when taking nitrates simultaneously, there will be a decrease in headaches and heart pain;
if you use Validol with glucose, it is possible that the pressure will increase slightly;
“Validol” for high blood pressure, taken together with drugs that have a calming effect on the nervous system, will help you fall asleep peacefully;
combined use with drugs that lower blood pressure will help enhance this effect.

“Validol” with glucose can be consumed, but only after consulting a specialist.

Cases of overdose

An overdose of Validol entails various negative consequences. Therefore, it is important to know how to take Validol correctly.

List of these phenomena:

Validol with glucose can cause an increase in blood sugar;
an overdose of Validol in some cases causes dizziness and migraines;
possible distortion of the heart;
decreased blood pressure;
negative effect on the central nervous system;
allergic manifestations.

If these cases occur, you should rinse your stomach.

Analogs

In the modern pharmaceutical industry there are many analogues of Validol.

Its substitutes are:

Substitutes for the drug have the same effect and have virtually no differences from the original. Analogues of Validol may differ only in price.