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Valerian extract and tablets. Valerian extract. Useful qualities

To calm the nervous system and normalize sleep, valerian extract in tablets is prescribed. Instructions for using the popular sedative are outlined in this post. Official name— Valerian extract film-coated tablets, […]

To calm the nervous system and normalize sleep, valerian extract in tablets is prescribed. Instructions for using the popular sedative are outlined in this post. The official name is Valerian extract film-coated tablets, 0.02 g, Latin version - Tabulettae Extracti Valerianae obductae 0.02 g.

Composition of yellow valerian tablets

Active ingredient in tablets

One yellow tablet contains 20 mg of the active substance, it is presented thick extract valerian plants.

Excipients in tablets

The drug also contains additional components, we list them below:

How many valerian tablets are in one package?

For the convenience of consumers, preparations containing 10, 20 and 50 coated tablets are produced. Typically, yellow tablets come in a glass bottle under a plastic cap. A small bottle is packed in cardboard box, it contains instructions. Valerian is also sold in cell packaging.

Indications for valerian tablets

Most often, valerian is used to correct conditions for these disorders:

vegetative-vascular dystonia ( incorrect operation autonomic nervous system, manifested by a whole spectrum of ailments),
excessive nervous excitability,
insomnia,
headache in the form of a migraine,
functional disorders in the cardiovascular system,
gastrointestinal spasms.

As a rule, valerian is taken as part of complex therapy.

Effect of valerian tablets on humans

Properties of valerian

It is known that the drug in tablets:

has a sedative effect,
eliminates increased anxiety,
makes it easier to fall asleep,
improves sleep quality.

This is what happens in the body under the influence of active phyto-substances:

inhibition of certain centers of the nervous system,
vasodilatation,
slow heartbeat,
relaxation of muscles in the digestive and urinary system.

With long courses, in addition to the listed actions, the following are observed:

copious secretion of bile,
drop in blood pressure.

Pharmacological effect of valerian

When taking the drug orally plant origin noted sedative effect, it is usually expressed moderately. The tablets help you fall asleep easily.

A significant role in the effect of valerian on the body is played by the presence of a special essential oil, consisting of:

isovaleric acid,
borneol.

In addition, a mild sedative effect occurs due to alkaloids and valepotriates, for example:

Khotenin,
valerine

Observing patients taking valerian, one can notice a slow increase in the sedative effect, over time it manifests itself stably.

How much do valerian tablets cost?

The well-known yellow coated tablets can be purchased at an affordable price. A herbal preparation without additives costs from 40 to 60 rubles, depending on the region.

How is valerian extract taken?

It is better to use any medications strictly according to the recommendations of the manufacturer or attending physician, without deviating from the prescribed doses. Usually good effect gives a proven regimen, according to which you need to take valerian 1-2 tablets three times a day, orally, after meals, with water. Before using valerian extract in tablets, the instructions for use should be carefully studied, as they contain important requirements for consumer safety.

One of our site visitors believes that you need to take Valerian tablets (20 mg) according to the following regimen: take 2 tablets 4 times a day for 6 weeks. This scheme was suggested to him by a pharmacist. Perhaps she is also correct. As you can see, the dosage regimen may be different. Therefore, it is advisable to take the drug as recommended by your doctor.

What are valerian tablets Evening?

Inexpensive pills are designed to improve sleep disorders. A harmonious combination of valerian root, peppermint oil and hops gives an excellent sedative effect, helps to get out of stress and improve heartbeat. Also biologically active additive Evening is available in the form of motherwort with valerian.

Valerian tablets for children

Experts prescribe valerian for children with:

Children under 1 year of age are prohibited from using any form of the drug. Drops are given as many drops as the child is old, diluted with water. For tablets there are the following frames:

children 3-5 years old - half a tablet three times a day,
children 5-7 years old - 1 tablet no more than 3 times a day.

In all cases, take half an hour before meals. Valerian is also used in children in the form of phytopackets.

Valerian tablets during pregnancy

It is not advisable for pregnant women to take valerian. This is done according to indications and under the supervision of a doctor. IN best case scenario From the tablets you can get:

sedative effect,
lowering blood pressure,
relieving uterine hypertonicity.

True, the drug always acts after some time; there is a so-called cumulative effect. A course lasting at least 1 month is required. The tablets are taken after meals, twice or thrice a day. Possible side effects, therefore, a problematic pregnancy can be included in the list of contraindications.

Valerian tablets for breastfeeding

Indications for the use of valerian for breastfeeding

Typically, nursing mothers resort to valerian for:

sleep disorders,
nervousness,
headaches due to stress,
depressive states,
loss of strength, general decrease in tone,
disruptions in the gastrointestinal tract,
feelings of anxiety and fear,
tachycardia, arrhythmias.

In any case, you should not take valerian tablets during breastfeeding without consulting a doctor. The doctor will help you choose the dosage and protect yourself from side effects.

How does valerian act on breastfeeding women?

In most cases, women are satisfied with the effect of valerian. If you take these pills correctly and monitor yourself and your child, you will notice the following positive changes:

sleep improves, insomnia disappears,
anxiety decreases, signs of stress decrease,
are expanding coronary vessels,
pressure decreases,
spasms are relieved.

Overdose of valerian in women during breastfeeding

Symptoms of overdose or individual intolerance in women during lactation are the same as in other cases:

constipation and itching;
nausea, vomiting,
increased blood pressure,
overexcitation of the central nervous system,
sleep disorders.

How does valerian act on infants?

At best, valerian has no effect on the child; at worst, he has an allergic reaction, which manifests itself as hives. The redness of the skin and itching bother me. Stomach upsets and increased gas formation, lethargy or overexcitement.

How to replace valerian in tablets for breastfeeding?

Alcohol tincture is not suitable for women with breastfeeding, it is better to use tablets or herbal decoction. You can also place the herb in your pillow or place it on your windowsill. This aromatherapy is beneficial for mother and child. Sometimes it is advisable for nursing mothers to take instead of valerian:

motherwort preparations,
Persen,
Tenoten,
Glycine,
Novo-Passit.

Features of taking valerian during lactation

If a mother plans her day incorrectly, does not have the support of relatives, cannot allocate time for rest, or simply does not know how to properly relieve stress, then caring for a newborn baby is associated with lack of sleep, chronic fatigue, increased irritability, constant drowsiness or insomnia. When choosing sedatives It is worth paying attention that many substances penetrate into breast milk, which means they fall into children's body. In this regard, valerian tablets are considered relatively safe.

Valerian often helps nursing mothers cope with postpartum depression and balances the condition. True, you should not completely rely only on pills. In case of constant fatigue and lack of sleep, you need to act comprehensively - involve relatives in caring for the child, look for suitable relaxation methods. For example, it is useful for women during pregnancy and lactation to practice yoga. If the body is exhausted, then in addition to sedatives, you need to take vitamin and mineral supplements. complex drug. Below is a photo of valerian tablets.

Valerian (extract in tablets): sedative herbal drug

Contraindications for Valerian tablets

It is believed that you should not drink valerian:

in the first trimester of pregnancy,
with fructose intolerance,
children under 1-3 years old (according to various sources),
people with a lack of sucrase and lactase enzymes in the body.

Contraindications include the state of glucose-galactose malabsorption. You should not take pills if an individual intolerance has been identified; it manifests itself in the form of an allergy to this particular drug. For example, sneezing and coughing, watery eyes, itchy skin and rashes on the body may bother you.

According to official instructions, the main contraindication is hypersensitivity to the components of the drug.

Possible harm of valerian tablets

The over-the-counter drug must be used with extreme caution. You can seriously harm your body if you self-medicate, take pills for too long a course, or constantly exceed the generally accepted dosage. In particular, there may be:

Most often, the drug causes harm if it is used incorrectly and contraindications are not followed.

Side effects when taking valerian tablets

The above-mentioned harmful aspects may occur when taking medications indiscriminately. There is also a range of side effects that are often detected even with the correct use of the drug. These include:

constant debilitating drowsiness,
severe decrease in muscle tone,
low ability to work,
slower thinking and speech,
various problems with stool, for example, with a long course, constipation is possible.

We also note that even if you follow the rules for taking valerian, the reaction normally slows down. First of all, those people who engage in particularly dangerous activities that require extreme concentration of attention should be careful. The same applies to drivers.

If you experience any discomfort, you should stop drinking valerian and contact your doctor to find out the reasons or change the drug.

What to do if you overdose on valerian tablets?

If a person is in under stress has significantly exceeded the dose, then instead of the desired calm, he begins to suffer from:

diarrhea or constipation,
nausea.

The following phenomena may also be of concern:

pronounced apathy towards everything,
dizziness,
red spots on the face,
dilated pupils,
increased blood pressure.

With an overdose of valerian drops, similar symptoms include exacerbation of gastrointestinal diseases, migraine headaches, constant nausea and heartburn, irregular heartbeat. If you suspect an overdose, you should immediately call ambulance, that is, dial 03 and explain the essence of the problem. In this case, immediately stop consuming valerian tablets. While waiting for a doctor to examine you, you need to induce vomiting in the victim. This can be achieved by drinking a large volume of water, bending slightly and placing 2 fingers deep into the oropharynx, right up to the small tongue.

Effect of valerian tablets on cats

Domestic cats may behave inappropriately near valerian preparations, which is explained specific action components of a plant on an animal's body. Instead of a mild sedative effect like in humans, cats experience euphoria. The thing is that the aroma of the plant strongly reminds them of the smell of pheromones that are part of cat urine. Under the influence of these substances, the emotional and hormonal background animals.

The nervous system of cats begins to work in a special way, the perception of reality is distorted, that’s where inappropriate behavior. Under the narcotic effect of valerian, animals begin to:

run away from imaginary opponents and chase them,
roll on the floor
tear curtains and wallpaper,
howl frighteningly
urinate in inappropriate places.

This effect appears almost immediately after taking the drugs. If a breeder offers an animal a valerian preparation in the form of an alcohol tincture, then he may soon encounter cat alcoholism and all the ensuing consequences, such as peptic ulcer, liver disease, kidney failure.

Valerian tincture may be harmful to animals. Valerian tablets are even worse. Everything is explained by the fact that the tablets are represented not only by plant materials. They contain only a quarter plant extract of the total mass of pills. It also contains the above-mentioned excipients of synthetic origin, to which the animal’s body can react with severe allergies. If after several minutes of euphoria the cat begins to deep dream and it is impossible to wake her up, you need to take her to the veterinary clinic immediately.

The reaction to the drug is different for all cats, so it has not yet been determined lethal dose. In any case, if an animal finds and accidentally consumes a large amount of medication in any form, it will have to be treated by a veterinarian.

Valerian does not kill cats in all cases. In exceptional cases in individually are appointed small doses for the following problems:

heart failure,
spasms in the gastrointestinal tract.

The drug is prescribed only by a doctor and exclusively in liquid form. It has been noticed that not all cats react with euphoria to valerian, some ignore it, some are frightened by the smell and cannot stand it. For example, Siamese cats As a rule, they do not perceive the aroma of valerian at all.

Interaction of valerian with other substances

Valerian with other medicines

It has been noticed that valerian tablets interact in a special way with some drugs, for example, it gives:

enhanced effect sleeping pills,
enhanced effect sedatives,
enhancing the effect of antispasmodics.

Valerian with alcohol

It is important to know that combining valerian and alcohol is inadmissible. In combination with ethyl alcohol the drug has a pronounced depression of the central nervous system. As a result, all reactions will be greatly slowed down in a person, he will become not just lethargic, but clearly inhibited. Difficulties with concentrating and understanding others, and disturbances in the motor sphere are expected.

Valerian tablets and alcohol tincture- definitely not compatible with alcoholic drinks. Valerian is mainly prescribed for psychoses and neuroses; in these conditions it is extremely dangerous to take alcohol. If you take these substances together, you can lose control of yourself, harm your health and lose your ability to work the next day.

How to store valerian tablets?

Like all medicines, valerian should be kept in a place where small children have no access. The optimal storage temperature is up to +15 degrees Celsius. The first aid kit should be dry and the packaging should be tightly closed. You can take the drug orally until the expiration date. You must carefully read the attached instructions and keep them with the tablets. It is better to keep them while using any medicines. original packaging, it contains the release date and expiration date information, which is why this is important.

In order for valerian extract in tablets to work correctly, the instructions for use must be read, but the question of the duration of the course must still be discussed with your doctor. These frames different people may vary depending on the body’s reaction to the drug and other individual characteristics.

For many years, the demand for valerian in the form of tinctures and tablets has not decreased, despite the fact that many attribute a placebo effect to these drugs and today there are more modern and effective sedatives.

Most widely used in folk and official medicine. It was used for treatment back in Ancient Greece. Modern pharmacology produces various drugs based on it, including valerian tinctures, extracts, teas that do an excellent job with nervous disorders and diseases of cardio-vascular system.

Chemical composition of the plant

The stems and rhizomes of the plant contain a huge amount useful substances. These are polysaccharides, a multiple list of organic acids - among them are malic, formic, acetic, palmitic and others. In addition, valerian contains a unique essential oil, which includes valerian-borneol ester, isovaleric acid, proazulene and other substances.

Beneficial properties of valerian

This plant has excellent antispasmodic, tonic and choleretic effect. A drug such as valerian extract can reduce the excitability of the nervous system and increase secretion gastric tract, relax smooth muscles and dilate coronary vessels. It is used as the main aid for many diseases. Diseases such as hypertension, migraine, tachycardia, epilepsy are among the ailments in which this medicinal plant is an indispensable tool. has strong sedative properties and is indicated for insomnia, hysteria, and nervous excitability. This drug is also indispensable for women’s health in menopause. The importance of valerian in the treatment of diseases is no less important. digestive system.

Preparations from the valerian plant

For medicinal purposes, the roots of the plant are harvested, most favorable time For their collection it is the end of summer-beginning of autumn. Aqueous and alcohol infusions, soothing teas, it is included in many medicines. Amazing properties has valerian extract. The price of this drug is low, but its effectiveness is high. In addition, the grass will an excellent remedy for taking baths, such procedures will help you completely relax and restore strength.

Contraindications

However, we should not forget that valerian extract has contraindications. It is important to comply correct dosage drug, since incorrect administration and long-term use lead to constant drowsiness, decreased performance and the appearance depressive state. You should not take the drug uncontrollably in old age, especially if there is a threat of stroke or heart attack, as well as chronic enterocolitis, in the first three months of pregnancy and in case of individual intolerance. In case of nausea, tachycardia, various allergic reactions, lethargy should stop taking valerian extract. It is also not recommended to use this remedy when driving a car or doing work that requires concentration.

LSR-005899/08

Tradename: Valerian extract

Dosage form:

film-coated tablets

Composition per tablet:

Active substance:
Valerian extract thick	– 0.02 g
Excipients:
magnesium carbonate basic (magnesium hydroxycarbonate), potato starch, croscarmellose sodium (primelose), calcium stearic acid (calcium stearate), gelatin	– sufficient quantity until received uncoated tablets weighing 0.1 g
Shell composition:
sugar (sucrose), basic magnesium carbonate (magnesium hydroxycarbonate), aerosil A-380 (colloidal silicon dioxide), titanium dioxide (titanium dioxide), gelatin, beeswax, tropeolin-O	– sufficient amount to receive the tablet, coated by extension method, weighing 0.20 g

Description
Biconvex, film-coated tablets yellow color.

Pharmacotherapeutic group
Sedative of plant origin.

ATX Code: N05CM09

pharmachologic effect
The active principle of the drug is the ester of borneol and isovaleric acid. It has a moderate sedative effect, which occurs slowly, but is quite stable. In addition, the drug has an antispasmodic effect on the smooth muscles of the gastrointestinal tract.

Indications for use
Increased nervous excitability, insomnia, functional disorders cardiovascular system, spasms of the gastrointestinal tract.

Contraindications
Hypersensitivity to the components of the drug, childhood up to 12 years old.
With caution - chronic enterocolitis.

Directions for use and doses
Take 1-2 tablets orally 3 times a day after meals.

Side effect
Possible lethargy, weakness, drowsiness, decreased performance (especially when used in high doses ah), at long-term use– constipation. In some cases, allergic reactions may develop.

Interaction with other drugs
Enhances the effect of hypnotics and other drugs that depress the central nervous system nervous system, as well as antispasmodics.

special instructions
With long-term use in large doses a decrease in psychomotor reactions is possible, which should be taken into account when driving, working with machinery, etc.

Release form
Film-coated tablets.
10 or 50 tablets in blister packs made of aluminum foil. 2, 3, 4, 5 blister packs No. 10 or 1 blister pack No. 50 together with instructions for use are placed in a cardboard pack.
900 contour blister packs No. 10 or 240 contour blister packs No. 50 along with the same number of instructions for use are placed in cardboard boxes.

Storage conditions
In a dry place at a temperature of 12 to 15 °C.
Keep out of the reach of children.

Best before date
5 years. Do not use after the expiration date.

Conditions for dispensing from pharmacies
Over the counter.

Manufacturer/Organization accepting complaints from consumers:
JSC "Pharmcenter VILAR"
117216, Russia, Moscow, st. Grina, 7.

Instructions for medical use medicine

Valerian extract

Tradename

Valerian extract

International nonproprietary name

Dosage form

Film-coated tablets 0.02 g

One tablet contains

active substance - thick valerian extract - 0.02 g,

excipients: basic magnesium carbonate, potato starch, talc, gelatin,

shell composition: basic magnesium carbonate, beeswax, titanium dioxide pigment, quinoline yellow (E-104), sugar, talc, colloidal silicon dioxide, gelatin, sunflower oil, paraffin.

Description

Yellow film-coated tablets with a biconvex surface. The cross section shows two layers.

Pharmacotherapeutic group

Sleeping pills and sedatives other

PBX code N05CM09

Pharmacological properties

Pharmacokinetics

The pharmacokinetics of valerian has been poorly studied, which is due to the impossibility of accurate identification effective start drug. After oral administration

600 mg dry extract of valerian maximum concentration of valeric acid (one of the probable active ingredients) is achieved after 1-2 hours and is 0.9-2.3 ng/ml. The half-life of elimination is 1.1 ± 0.6 hours. With repeated use of the drug, its pharmacokinetics do not change.

Pharmacodynamics

Herbal remedy. Has a sedative effect.

The effect is due to the content of essential oil (0.2-2.8%), most of which is the ester of borneol and isovaleric acid - borneol acetate. Important components of the drug are also contained in the roots of valerian - sexviterpenes and monoterpenes: β-caryophyllene, valeranone, valeral, valeric acid, as well as valepotriates (0.05-0.67%) - valtrate and isovaltrate. The main degradation products of valepotriates are baldrinal, homobaldrinal and valtroxal. Valerian extract increases the sensitivity of GABA receptors (gamma-amino butyric acid receptors) to the effects of γ -aminobutyric acid, which enhances inhibition processes in the cerebral cortex. At the same time, an increase in the synthesis and secretion of GABA is observed at the synapses of neurons in the cerebral cortex. This effect manifests itself only under the influence of the sum of substances contained in the valerian extract and cannot be reproduced with the isolated administration of essential oil, sexviterpenes or valepotriates.

The sedative effect when using valerian appears slowly, but quite steadily and fully develops only with systematic and long-term course treatment. The speed of the body's reaction to external stimuli, the onset of natural sleep is facilitated.

Valepotriates and valeric acid have an antispasmodic effect and have a slight choleretic effect, especially in cases of spasm and hypermotor dyskinesia of the biliary tract.

Complex biologically active substances Valerian, through neurohumoral mechanisms and influences on the myocardial conduction system, regulates cardiac activity - slows down the heart rate, slightly dilates the coronary vessels.

Indications for use

neurasthenia and conditions associated with prolonged neuropsychic agitation

sleep disturbances due to overexcitation, nervous stress

mild functional disorders of the cardiovascular system and digestive system (as part of complex therapy).

Directions for use and doses

Adults: 40-80 mg (2-4 tablets) 3 times a day. If necessary daily dose can be increased to 1000 mg in several (usually 4-5) doses. In persons with impaired liver and kidney function, no dose adjustment is required.

The course of treatment is up to 1 month.

Side effects

Lethargy, depression, weakness, decreased performance

In some cases: allergic reactions may develop.

Contraindications

Hypersensitivity to valerian and excipients drug

Children and teenagers up to 18 years of age.

Drug interactions

Valerian potentiates the effect of other sedatives and hypnotics, anesthetics, psychotropic drugs, and antispasmodics.

special instructions

Pregnancy and lactation

Taking valerian extract during pregnancy does not have a teratogenic effect. Considering side effects the drug must be used with caution during lactation

Features of the effect of the drug on the ability to drive vehicle or potentially dangerous mechanisms

The lethargy and decreased response to external stimuli caused by valerian preparations, as a rule, does not affect the patient’s ability to drive a vehicle or other operator activities. However, caution is required, especially when combining valerian with alcohol-containing drinks or other drugs that affect the central nervous system.

Overdose

Symptoms: when using excessively high doses (more than 20 times the maximum recommended dose), nonspecific symptoms associated with depression of the central nervous system may occur: lethargy, lethargy, drowsiness. IN severe cases bradycardia and arrhythmia may occur.